Publications and projects

Grupo de Química Computacional (GQC), CEQUINOR (UNLP, CONICET), Facultad de Ciencias Exactas, Universidad Nacional de La Plata, Argentina.

Researcher profiles

Researcher Google Scholar Institutional profile
Reinaldo Pis Diez Scholar
Martín J. Lavecchia Scholar CEQUINOR, CONICET

Full institutional record: CEQUINOR publications and CONICET Digital.

Publications, 2022 to 2026

2026

KINOTECA: A Navigator of Chemical Datasets with Reported Kinase Inhibitory Activity Guarimata, J.D.; Martínez Heredia, L.; Montiel, E.; Quispe, P.A.; Lavecchia, M.J. Kinases Phosphatases 2026, 4, 22 DOI:10.3390/kinasesphosphatases4030022

Glycosyl coumarins as selective inhibitors of tumor-associated carbonic anhydrase IX and XII: synthesis, structure-activity relationships, and molecular modeling Le Pors, M. S.; Aznar, I.; Giovannuzzi, S.; Supuran, C. T.; Lavecchia, M. J.; Colinas, P. A. International Journal of Molecular Sciences 2026, 27 (8), 3659. DOI: 10.3390/ijms27083659

2025

A critical assessment of computer-aided approaches for identifying FAK inhibitors Quispe-Castillo, P. A.; Lietha, D.; León, I. E.; Lavecchia, M. J. Kinases and Phosphatases 2025, 3 (4), 27. DOI: 10.3390/kinasesphosphatases3040027

NaturAr: a collaborative, open-source database of natural products from Argentinian biodiversity for drug discovery and bioprospecting Martínez Heredia, L.; Quispe, P. A.; Fernández, J. F.; Lavecchia, M. J. Journal of Chemical Information and Modeling 2025, 65 (4), 1889-1900. DOI: 10.1021/acs.jcim.4c01507

Target Fisher: a consensus structure-based target prediction tool, and its application in the discovery of selective MAOB inhibitors Fernández, J. F.; Martínez Heredia, L.; Caracciolo, F.; Esses, D.; Suarez, R.; Siless, G.; Perez, C.; Rodríguez-Franco, M. I.; Fernández, L. R.; Palermo, J. A.; Lavecchia, M. J. Chemistry, a European Journal 2025, 31 (1). DOI: 10.1002/chem.202401838

Update and ADMET profile of the Latin American Natural Product Database: LANaPDB Gómez-García, A.; Lavecchia, M. J.; Olmedo, D. A.; Solís, P. N.; Medina-Franco, J. L. Molecular Informatics 2025, 44, e70013. DOI: 10.1002/minf.70013

Glucoimines incorporating classical and non-classical carbonic anhydrase pharmacophores: design, synthesis, conformational analysis, biological evaluation, and docking simulations Vásquez, I. R.; Riafrecha, L. E.; Martínez Heredia, L.; Echeverría, G. A.; Piro, O. E.; Lavecchia, M. J.; Supuran, C. T.; Colinas, P. A. Journal of Molecular Structure 2025, 1321, 139778. DOI: 10.1016/j.molstruc.2024.139778

Quantitative structure-property relationship for gas-chromatographic retention indices of volatile organic compounds in colored-quinoa seeds Rojas, C.; Cedillo, J. F.; Sarmiento, N.; Pis Diez, R.; Duchowicz, P. R. Journal of Food Composition and Analysis 2025, 137, 106843. DOI: 10.1016/j.jfca.2024.106843

2024

A computational study of the role of cobalt in thiophene adsorption on small Mo and MoCo clusters as site models for the HDS process Del Plá, J.; Pis Diez, R. Surface Science 2024, 749, 122571. DOI: 10.1016/j.susc.2024.122571

Computational prediction of retention times of veterinary antibiotics obtained by liquid chromatography-mass spectrometry Rojas, C.; Sarmiento, N.; Ayora, E.; Pis Diez, R. Journal of the Science of Food and Agriculture 2024. DOI: 10.1002/jsfa.13499

Structural and spectroscopic study and intermolecular chalcogen bonding interactions in 1,3-dicarbonyl compounds Vallejo, L. S.; Jios, J. L.; Ulic, S. E.; Echeverría, G. A.; Piro, O. E.; Pis Diez, R.; Vázquez, C.; Merlo, C. New Journal of Chemistry 2024, 48 (32), 14420-14434. DOI: 10.1039/D4NJ02508C

Unanticipated synthesis of a C3 symmetrical tris-triazine under cyclization conditions of coumarinoyl thioureas with alpha-halo compounds Shabir, G.; Ashraf, S.; Saeed, A.; Hashmi, M. Z.; Hökelek, T.; Nossa González, D. L.; Pis Diez, R.; El-Seedi, H. R.; Bolte, M.; Erben, M. F. Journal of Molecular Structure 2024, 1304, 137686. DOI: 10.1016/j.molstruc.2024.137686

Exploring the potential anti-thyroid activity of acetyl-L-carnitine: lactoperoxidase inhibition profile, iodine complexation and scavenging power against H2O2. Experimental and theoretical studies Caro-Ramírez, J. Y.; Franca, C. A.; Lavecchia, M. J.; Naso, L. G.; Williams, P. A. M.; Ferrer, E. G. Spectrochimica Acta Part A: Molecular and Biomolecular Spectroscopy 2024, 313, 124098. DOI: 10.1016/j.saa.2024.124098

Alkaline phosphatase inhibition and antithyroid activity of an acetylacetone sulfonamide derived Schiff base. In vitro and in silico studies Gaddi, G. M.; Caro-Ramírez, J. Y.; Antonena, Y. B.; Franca, C. A.; Martínez Heredia, L.; Lavecchia, M. J.; Williams, P. A. M.; Ferrer, E. G. ChemistrySelect 2024, 9 (23), e202401342. DOI: 10.1002/slct.202401342

Synthesis and supramolecular behaviour study of a novel amphiphilic compound for idebenone encapsulation Costantino, M. L. B.; Lavecchia, M. J.; Fascio, M. L.; Lastra, M. L.; Contin, M. D.; D'Accorso, N. B. Journal of Molecular Structure 2024, 137936. DOI:

Drug interaction profiles classification: Sørensen-Dice coefficient based on MM/GBSA energies to explore focal adhesion kinase inhibitors Quispe, P. A.; Martínez Heredia, L.; León, I. E.; Lavecchia, M. J. ChemRxiv 2024, preprint. DOI: 10.26434/chemrxiv-2024-jzk7n

2023

Chemoinformatic modelling of the antioxidant activity of phenolic compounds Idrovo-Encalada, A. M.; Rojas, A. M.; Fissore, E. N.; Tripaldi, P.; Pis Diez, R.; Rojas, C. Journal of the Science of Food and Agriculture 2023, 103 (10), 4867-4875. DOI: 10.1002/jsfa.12561

Novel fluoroquinolones with possible antibacterial activity in Gram-negative resistant pathogens: in silico drug discovery Coba-Males, M. A.; Lavecchia, M. J.; Alcívar-León, C. D.; Santamaría-Aguirre, J. Molecules 2023, 28 (19), 6929. DOI: 10.3390/molecules28196929

Molecular docking for the development of alternative therapies against leishmaniasis Guarimata, J. D.; Alcívar-León, C. D.; Lavecchia, M. J.; Poveda, A. Chemistry Proceedings 2023, 14 (1), 82. DOI: 10.3390/ecsoc-27-16050

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